Delaware
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11-3516358
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(State or other jurisdiction of incorporation or organization)
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(I.R.S. Employer Identification Number)
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Large Accelerated Filer
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o
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Accelerated Filer
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þ
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Non-Accelerated Filer
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o
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Smaller reporting company
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o
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(Do not check if a smaller reporting company)
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Page
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PART I
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FINANCIAL INFORMATION
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Item 1
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Financial Statements
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1)
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3
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2)
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4
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3)
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5
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4)
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7
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Item 2
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38
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Item 3
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47
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Item 4
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47
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PART II
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OTHER INFORMATION
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|||
Item 1
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48
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|||
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||||
Item 1A
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48
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|||
Item 2
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48
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Item 3
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48
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Item 4
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48
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Item 5
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48
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Item 6
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48
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49
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September 30, 2011
(unaudited)
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December 31,
2010
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|||||||
ASSETS
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||||||||
Current Assets:
|
||||||||
Cash and cash equivalents
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$ | 13,216,933 | $ | 12,340,239 | ||||
Marketable securities (note 4)
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1,950,000 | 2,451,620 | ||||||
Research tax credit receivable
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- | 145,513 | ||||||
Prepaid expenses and other current assets (note 5)
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455,709 | 706,649 | ||||||
Note receivable – current portion (note 6)
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25,688 | 28,023 | ||||||
Total Current Assets
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15,648,330 | 15,672,044 | ||||||
Restricted Cash Equivalents (note 18)
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2,947,451 | 401,893 | ||||||
Note Receivable (note 6)
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- | 18,682 | ||||||
Equipment, Net (note 7)
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93,072 | 123,565 | ||||||
Total Assets
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$ | 18,688,853 | $ | 16,216,184 | ||||
LIABILITIES AND STOCKHOLDERS’ EQUITY
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||||||||
Current Liabilities:
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||||||||
Accounts payable and accrued expenses (note 8)
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$ | 3,905,460 | $ | 1,820,900 | ||||
Deferred Research and Development Arrangement (note 9)
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843,750 | 900,000 | ||||||
Other Liabilities (note 10)
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113,640 | 133,117 | ||||||
Warrant Liabilities (note 15)
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3,653,706 | 2,966,710 | ||||||
Total Liabilities
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8,516,556 | 5,820,727 | ||||||
Commitments and Contingencies (note 18)
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||||||||
Stockholders’ Equity (note 13):
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||||||||
Preferred stock, par value $0.0001, 100,000,000 authorized shares, none issued and outstanding
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- | - | ||||||
Common stock, par value $0.0001, 500,000,000 authorized shares, 95,279,861 (2010 – 84,175,504) issued and 95,265,656 (2010 – 84,160,849) outstanding
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9,528 | 8,418 | ||||||
Additional paid-in capital
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67,665,073 | 56,157,452 | ||||||
Accumulated other comprehensive loss
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- | (2,340 | ) | |||||
Accumulated deficit during the development stage
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(57,473,894 | ) | (45,739,663 | ) | ||||
Treasury stock, 14,205 shares, at cost
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(28,410 | ) | (28,410 | ) | ||||
Total Stockholders’ Equity
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10,172,297 | 10,395,457 | ||||||
Total Liabilities and Stockholders’ Equity
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$ | 18,688,853 | $ | 16,216,184 |
For the Three Months Ended
September 30,
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For the Nine Months Ended
September 30,
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Cumulative
from March 19, 2001
(Inception) to
September 30,
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||||||||||||||||||
2011
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2010
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2011
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2010
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2011
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||||||||||||||||
(Restated)
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(Restated)
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|||||||||||||||||||
Revenues:
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||||||||||||||||||||
Research
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$ | - | $ | - | $ | - | $ | - | $ | - | ||||||||||
Expenses:
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||||||||||||||||||||
General and administrative
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774,307 | 1,561,377 | 2,811,097 | 4,423,376 | 26,610,263 | |||||||||||||||
Research and development
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2,372,201 | 671,339 | 10,506,823 | 2,453,350 | 30,400,339 | |||||||||||||||
Patent fees
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198,424 | 123,147 | 374,163 | 238,089 | 1,929,141 | |||||||||||||||
Depreciation and amortization
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10,127 | 11,663 | 34,904 | 34,843 | 630,371 | |||||||||||||||
Total Expenses
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3,355,059 | 2,367,526 | 13,726,987 | 7,149,658 | 59,570,114 | |||||||||||||||
Loss from Operations
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(3,355,059 | ) | (2,367,526 | ) | (13,726,987 | ) | (7,149,658 | ) | (59,570,114 | ) | ||||||||||
Other Income (Expense)
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||||||||||||||||||||
Realized loss on marketable securities .
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- | - | (3,960 | ) | - | (13,301 | ) | |||||||||||||
Interest income
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19,592 | 49,418 | 100,914 | 97,699 | 1,412,981 | |||||||||||||||
Interest expense
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- | - | - | - | (301,147 | ) | ||||||||||||||
Other income
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- | - | - | 56,047 | 56,047 | |||||||||||||||
Unrealized gain (loss) on fair value of warrants
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1,866,249 | 2,536,999 | 1,993,469 | (4,333,496 | ) | 891,124 | ||||||||||||||
Unrealized gain on fair value of put feature on common stock
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- | - | - | 97,713 | 2,315,539 | |||||||||||||||
Financing expense
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- | - | (97,667 | ) | (180,080 | ) | (640,023 | ) | ||||||||||||
Beneficial conversion feature
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- | - | - | - | (1,625,000 | ) | ||||||||||||||
Total Other Income (Expense)
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1,885,841 | 2,586,417 | 1,992,756 | (4,262,117 | ) | 2,096,220 | ||||||||||||||
Net (Loss) Income Before Provision for Income Taxes
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(1,469,218 | ) | 218,891 | (11,734,231 | ) | (11,411,775 | ) | (57,473,894 | ) | |||||||||||
Provision for income taxes
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- | - | - | - | - | |||||||||||||||
Net (Loss) Income
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$ | (1,469,218 | ) | $ | 218,891 | $ | (11,734,231 | ) | $ | (11,411,775 | ) | $ | (57,473,894 | ) | ||||||
Net loss per share, basic and diluted
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$ | (0.02 | ) | $ | 0.00 | $ | (0.13 | ) | $ | (0.15 | ) | |||||||||
Weighted average number of shares outstanding, basic and diluted
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95,240,221 | 83,063,250 | 92,276,111 | 76,932,814 |
For the Nine Months Ended
September 30,
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Cumulative
From March 19, 2001
(Inception) to
September 30,
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|||||||||||
2011
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2010
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2011
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||||||||||
(Restated)
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||||||||||||
Cash Flows from Operating Activities:
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||||||||||||
Net loss
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$ | (11,734,231 | ) | $ | (11,411,775 | ) | $ | (57,473,894 | ) | |||
Adjustments to reconcile net loss to net cash used in operating activities:
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||||||||||||
Beneficial conversion feature
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- | - | 1,625,000 | |||||||||
Compensatory stock
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- | 1,663,999 | 2,129,877 | |||||||||
Depreciation and amortization
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34,904 | 34,843 | 630,371 | |||||||||
Stock-based compensation
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513,255 | 435,305 | 5,452,277 | |||||||||
Amortization of deferred research and development contribution
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(56,250 | ) | (56,250 | ) | (656,250 | ) | ||||||
Note receivable
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21,017 | (53,711 | ) | (25,688 | ) | |||||||
Realized losses on marketable securities
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3,960 | - | 13,301 | |||||||||
Unrealized (gain) loss on fair value of warrants
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(1,993,469 | ) | 4,333,496 | (891,124 | ) | |||||||
Unrealized gain on fair value of put feature on common stock
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- | (97,713 | ) | (2,315,539 | ) | |||||||
Financing expense
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97,667 | 180,080 | 640,023 | |||||||||
Amortization of deferred lease incentive
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(15,000 | ) | (15,000 | ) | (45,000 | ) | ||||||
Deferred lease expenses
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(4,477 | ) | 24,728 | 58,640 | ||||||||
Loss on impairment of intangible assets
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- | - | 286,132 | |||||||||
Changes in assets and liabilities:
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||||||||||||
Prepaid expenses and other current assets
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250,940 | (160,113 | ) | (455,709 | ) | |||||||
Research tax credit receivable
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145,513 | - | - | |||||||||
Accounts payable and accrued expenses
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2,084,560 | 555,268 | 3,905,460 | |||||||||
Net Cash Used in Operating Activities
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(10,651,611 | ) | (4,566,843 | ) | (47,122,123 | ) | ||||||
Cash Flows from Investing Activities:
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||||||||||||
Restricted cash equivalents
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(2,545,558 | ) | 842,454 | (2,947,451 | ) | |||||||
Purchase of equipment
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(4,411 | ) | (3,744 | ) | (553,359 | ) | ||||||
Purchase of marketable securities
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(8,000,000 | ) | (503,960 | ) | (21,123,960 | ) | ||||||
Proceeds from sales of marketable securities
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8,500,000 | 75,000 | 19,160,659 | |||||||||
Payment of licensing fees
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- | - | (356,216 | ) | ||||||||
Net Cash (Used in) Provided by Investing Activities
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(2,049,969 | ) | 409,750 | (5,820,327 | ) | |||||||
Cash Flows from Financing Activities:
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||||||||||||
Issuance of common stock and units, net of issuance costs
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13,220,273 | 9,318,228 | 55,805,574 | |||||||||
Proceeds from exercise of stock options
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40,040 | 107,240 | 150,882 | |||||||||
Proceeds from exercise of stock warrants
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317,961 | 3,263,376 | 3,581,337 | |||||||||
Proceeds from long-term debt
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- | - | 5,150,000 | |||||||||
Proceeds from research contribution
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- | - | 1,500,000 | |||||||||
Purchase of treasury stock
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- | - | (28,410 | ) | ||||||||
Net Cash Provided by Financing Activities
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13,578,274 | 12,688,844 | 66,159,383 | |||||||||
Net Increase in Cash and Cash Equivalents
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876,694 | 8,531,751 | 13,216,933 | |||||||||
Cash and Cash Equivalents – beginning of period
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12,340,239 | 7,298,032 | - | |||||||||
Cash and Cash Equivalents - end of period
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$ | 13,216,933 | $ | 15,829,783 | $ | 13,216,933 |
For the Nine Months Ended
September 30,
|
Cumulative
From March 19, 2001
(Inception) to
September 30,
|
|||||||||||
2011
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2010
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2011
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||||||||||
(Restated)
|
||||||||||||
Supplemental Cash Flow Information
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||||||||||||
Interest paid
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$ | - | $ | - | $ | 301,147 | ||||||
Non-cash financing and investing activities:
|
||||||||||||
Warrants issued
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$ | 2,924,333 | $ | 1,980,880 | $ | 11,054,427 | ||||||
Put feature on common stock issued
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$ | - | $ | - | $ | 4,954,738 | ||||||
Dilutive issuances of common stock
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$ | - | $ | - | $ | 2,639,199 | ||||||
Warrant liability extinguishment from exercise of warrants
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$ | 243,868 | $ | 5,286,602 | $ | 6,180,660 | ||||||
Leasehold improvement incentive
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$ | - | $ | - | $ | 100,000 | ||||||
Settlement of lawsuit
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$ | - | $ | 43,953 | $ | 43,953 |
1.
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Operations and Organization
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2.
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Prior Period Adjustment
|
STATEMENT OF OPERATIONS FOR THE THREE MONTHS ENDED SEPTEMBER 30, 2010
|
||||||||||||
As previously reported
|
Effect of Restatement
|
As restated
|
||||||||||
Unrealized gain on fair value of warrants
|
- | 2,536,999 | 2,536,999 | |||||||||
Total other income (expense)
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49,418 | 2,536,999 | 2,536,999 | |||||||||
Net (loss) income before provision for income taxes
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(2,318,108 | ) | 2,536,999 | 218,891 | ||||||||
Net (loss) income
|
(2,318,108 | ) | 2,536,999 | 218,891 | ||||||||
Net (loss) income per share, basic and diluted
|
(0.03 | ) | 0.03 | 0.00 |
STATEMENT OF OPERATIONS FOR THE NINE MONTHS ENDED SEPTEMBER 30, 2010
|
||||||||||||
As previously reported
|
Effect of Restatement
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As restated
|
||||||||||
Unrealized gain on fair value of put feature on common stock
|
- | 97,713 | 97,713 | |||||||||
Unrealized loss on fair value of warrants
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- | (4,333,496 | ) | (4,333,496 | ) | |||||||
Financing expense
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- | (180,080 | ) | (180,080 | ) | |||||||
Total other income (expense)
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153,746 | (4,415,863 | ) | (4,262,117 | ) | |||||||
Net loss before provision for income taxes
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(6,995,912 | ) | (4,415,863 | ) | (11,411,775 | ) | ||||||
Net loss
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(6,995,912 | ) | (4,415,863 | ) | (11,411,775 | ) | ||||||
Net loss per share, basic and diluted
|
(0.09 | ) | (0.06 | ) | (0.15 | ) |
2.
|
Prior Period Adjustment (cont’d)
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STATEMENT OF CASH FLOWS FOR THE NINE MONTHS ENDED SEPTEMBER 30, 2010
|
||||||||||||
As previously reported
|
Effect of Restatement
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As restated
|
||||||||||
Net loss
|
(6,995,912 | ) | (4,415,863 | ) | (11,411,775 | ) | ||||||
Unrealized gain on fair value of put feature on common stock
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- | (97,713 | ) | (97,713 | ) | |||||||
Unrealized loss on fair value of warrants
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- | 4,333,496 | 4,333,496 | |||||||||
Financing expense
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- | 180,080 | 180,080 | |||||||||
Net cash used in operating activities
|
(4,566,843 | ) | - | (4,566,843 | ) |
3.
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Recent Accounting Pronouncements Affecting the Company
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4.
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Marketable Securities
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Securities available-for-sale
|
Cost
Basis |
Gross
Unrealized
Losses |
Fair
Value |
|||||||||
September 30, 2011:
|
||||||||||||
State and municipal obligations
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$ | 1,950,000 | $ | - | $ | 1,950,000 | ||||||
December 31, 2010:
|
||||||||||||
State and municipal obligations
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$ | 2,453,960 | $ | (2,340 | ) | $ | 2,451,620 |
Maturity
|
Cost
Basis |
Gross
Unrealized
Losses |
Fair
Value |
|||||||||
10 years or more
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$ | 1,950,000 | - | $ | 1,950,000 |
5.
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Prepaid Expenses and Other Current Assets
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September 30,
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December 31,
|
|||||||
2011
|
2010
|
|||||||
Deposits on contracts
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$ | 244,131 | $ | 564,074 | ||||
Other assets
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211,578 | 142,575 | ||||||
$ | 455,709 | $ | 706,649 |
6.
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Note Receivable
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Principal Amortization
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Expected
Payment
|
|||
Within 1 year
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$ | 25,688 |
7.
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Equipment, Net
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September 30,
2011
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December 31,
2010
|
|||||||
Furniture and fixtures
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$ | 32,646 | $ | 32,169 | ||||
Office equipment
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80,120 | 77,032 | ||||||
Lab and computer equipment
|
430,261 | 429,415 | ||||||
Leasehold improvements
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110,713 | 110,713 | ||||||
Total fixed assets
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653,740 | 649,329 | ||||||
Less: Accumulated depreciation
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(560,668 | ) | (525,764 | ) | ||||
Net carrying amount
|
$ | 93,072 | $ | 123,565 |
8.
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Accounts Payable and Accrued Expenses
|
September 30,
2011
|
December 31,
2010
|
|||||||
Trade payables
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$ | 2,039,922 | $ | 489,527 | ||||
Accrued expenses
|
25,400 | 18,466 | ||||||
Accrued research and development contract costs
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1,706,650 | 1,239,233 | ||||||
Payroll liabilities
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133,488 | 73,674 | ||||||
$ | 3,905,460 | $ | 1,820,900 |
9.
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Deferred Research and Development Arrangement
|
10.
|
Other Liabilities
|
10.
|
Other Liabilities (cont’d)
|
September 30,
2011
|
December 31,
2010
|
|||||||
Deferred lease incentive
|
$ | 100,000 | $ | 100,000 | ||||
Less accumulated amortization
|
(45,000 | ) | (30,000 | ) | ||||
Balance
|
$ | 55,000 | $ | 70,000 |
11.
|
Comprehensive Loss
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12.
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Net Loss per Common Share
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13.
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Common Stock
|
|
a)
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On May 10, 2001, the Company issued 3,600,000 shares of common stock to the Company’s founders for cash of $1.
|
|
b)
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On August 10, 2001, the Company issued:
|
|
i)
|
1,208,332 shares of common stock to the directors of the Company for cash of $1,450,000.
|
|
ii)
|
958,334 shares of common stock to Rexgene for cash of $550,000.
|
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iii)
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360,000 shares of common stock in a private placement to individual investors for cash of $1,080,000.
|
|
c)
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On October 10, 2001, the Company issued 400,000 shares of common stock to Chong Kun Dang Pharmaceutical Corp. (“CKD”) for cash of $479,991 and 400,000 shares of common stock to an individual investor for cash of $479,991.
|
|
d)
|
On October 10, 2001, the Company issued 200,000 shares of common stock to CKD for cash of $479,985.
|
|
e)
|
Since inception, the Company’s founders have transferred 800,000 shares of the common stock described in a) to officers and directors of the Company.
|
|
f)
|
In July 2003, the stockholders described in b) (iii) and e) transferred an aggregate of 1,268,332 shares of common stock to a voting trust. The trust allows for the unified voting of the stock by the trustees.
|
|
g)
|
On August 20, 2003, the Company issued 500,000 shares of common stock to KT&G Corporation for cash consideration of $2,000,000.
|
|
h)
|
On October 29, 2004, an option holder exercised options to purchase shares of common stock for cash of $1,800 and the Company issued an aggregate of 1,500 shares.
|
|
i)
|
Pursuant to the agreement and plan of merger which occurred on May 13, 2005, (i) each share of the issued and outstanding common stock of Rexahn, Corp (“Rexahn”) (other than dissenting shares) was converted into the right to receive five shares of Rexahn Pharmaceuticals common stock; (ii) each issued, outstanding and unexercised option to purchase a share of Rexahn common stock was converted into an option to purchase five shares of Rexahn Pharmaceuticals’ common stock and (iii) the par value of Rexahn’s common stock was adjusted to reflect the par value of Corporate Road Show Com Inc. (“CRS”) common stock. In the acquisition merger, 289,780,000 CRS pre-reverse stock split shares were converted into 2,897,802 post-reverse stock split Rexahn Pharmaceuticals shares, and an additional 500,000 post-reverse stock split Rexahn Pharmaceuticals shares were issued to a former executive of CRS. All shares and earnings per share information have been retroactively restated in these financial statements.
|
|
j)
|
On August 8, 2005, the Company issued, in a transaction exempt from registration under the Securities Act of 1993, as amended, 4,175,000 shares of common stock at a purchase price of $2.00 per share.
|
|
k)
|
On October 3, 2005, the Company issued 7,000 shares of common stock for $21,877 and $7,500 cash in exchange for legal services from W. Rosenstadt and Steve Sanders.
|
13.
|
Common Stock (cont’d)
|
l)
|
On December 2, 2005, the holders of a convertible note that was issued on August 8, 2005 and, represented $1,300,000 aggregate principal amount, exercised their option to convert the entire principal amount of the note into the Company’s common stock. Based on a $2.00 per share conversion price, the holders received an aggregate of 650,000 shares.
|
m)
|
On December 27, 2005, option holders exercised options to purchase shares of the Company’s common stock for cash of $9,600 and the Company issued an aggregate of 40,000 shares.
|
n)
|
On February 22, 2006, an option holder exercised options to purchase shares of the Company’s common stock for cash of $1,200 and the Company issued an aggregate of 5,000 shares.
|
o)
|
On April 12, 2006, an option holder exercised options to purchase shares of the Company’s common stock for cash of $3,409 and the Company issued an aggregate of 14,205 shares. On the same date, the Company agreed to repurchase common stock from the option holder based on the then market price for treasury in exchange for the aggregate purchase price of $28,410 in cash.
|
p)
|
On May 13, 2006, holders of the $3,850,000 convertible notes issued on February 28, 2005, exercised their rights to convert the entire principal amount of the notes into shares of the Company’s common stock. Based on a $1.00 per share conversion price, the Company issued 3,850,000 shares of common stock in connection with the conversion.
|
q)
|
On October 9, 2006, an option holder exercised options to purchase shares of the Company’s common stock for cash of $2,400 and the Company issued an aggregate of 10,000 shares.
|
r)
|
On November 19, 2006, an option holder exercised options to purchase shares of the Company’s common stock for cash of $1,800 and the Company issued an aggregate of 7,500 shares.
|
s)
|
On December 19, 2006, an option holder exercised options to purchase shares of the Company’s common stock for cash of $6,000 and the Company issued an aggregate of 25,000 shares.
|
t)
|
On April 18, 2007, an option holder exercised options to purchase shares of the Company’s common stock for cash of $14,400 and the Company issued an aggregate of 18,000 shares.
|
u)
|
On July 23, 2007, an option holder exercised options to purchase shares of the Company’s common stock for cash of $12,000 and the Company issued an aggregate of 15,000 shares.
|
v)
|
On September 27, 2007, an option holder exercised options to purchase shares of the Company’s common stock for cash of $15,600 and the Company issued an aggregate of 19,500 shares.
|
13.
|
Common Stock (cont’d)
|
w)
|
On December 18, 2007, the Company issued 4,857,159 units at a price $1.40 per share for total gross proceeds of $6,800,023. Investors also were issued one warrant for every five shares purchased. One warrant will entitle the holder to purchase an additional share of common stock at a purchase price of $1.80 at any time over a period of three years from the date of the closing. The Company has recorded the warrants as liabilities at fair value as disclosed in Note 15. Private placement closing costs of $139,675 were recorded as a reduction of the issuance proceeds. Private placements costs also consist of 107,144 warrants, valued at $138,326, and were recorded as a financing expense. The Company extended anti-dilutive protection to the investors. The anti-dilution protection provision is structured in a way that is designed to protect a holder’s position from being diluted and contains a price protection based on a mathematical calculation, and is recorded as a liability at fair value, as disclosed in Note 16. The Company revalues these liabilities each reporting period, with the unrealized gain (loss) recorded as other income (expense).
|
Gross Proceeds:
|
$ | 6,800,023 | ||
Allocated to liabilities:
|
||||
Warrant liabilities
|
1,392,476 | |||
Put feature on common stock
|
4,401,169 | |||
Total allocated to liabilities
|
5,793,645 | |||
Allocated to equity:
|
||||
Common stock and additional paid-in capital
|
1,144,704 | |||
Allocated to expense:
|
||||
Financing expense
|
(138,326 | ) | ||
Total allocated gross proceeds:
|
$ | 6,800,023 |
x)
|
On December 27, 2007, an option holder exercised options to purchase shares of the Company’s common stock for cash of $18,000 and the Company issued an aggregate of 75,000 shares.
|
13.
|
Common Stock (cont’d)
|
y)
|
On March 20, 2008, the Company issued 642,858 units consisting of one share of the Company’s common stock and one warrant for every five common shares purchased in a private placement at a price of $1.40 per unit for total gross proceeds of $900,001. One warrant will entitle the holder to purchase an additional share of common stock at a price of $1.80 at any time over a period of three years from the date of the private placement, and is recorded as a liability at fair value. The Company extended anti-dilution protection to investors, and the provision is structured in a way that is designed to protect the holder’s position from being diluted and contains a price based on a mathematical computation.
|
Gross Proceeds:
|
$ | 900,001 | ||
Allocated to liabilities:
|
||||
Warrant liabilities
|
190,917 | |||
Put feature on common stock
|
553,569 | |||
Total allocated to liabilities
|
744,486 | |||
Allocated to common stock and additional paid-in capital
|
155,515 | |||
Total allocated gross proceeds:
|
$ | 900,001 |
z)
|
On May 30, 2008, an option holder exercised options to purchase shares of the Company’s common stock for cash of $7,200 and the Company issued an aggregate of 30,000 shares.
|
aa)
|
On June 2, 2008, an option holder exercised options to purchase shares of the Company’s common stock for cash of $12,000 and the Company issued an aggregate of 50,000 shares.
|
ab)
|
On June 30, 2008, an option holder exercised options to purchase shares of the Company’s common stock for cash of $12,000 and the Company issued an aggregate of 10,000 shares.
|
13.
|
Common Stock (cont’d)
|
ac)
|
On June 5, 2009 the Company closed on a purchase agreement to issue 2,857,143 shares of common stock at a price of $1.05 per share to an institutional investor for total gross proceeds of $3,000,000 and incurred $289,090 of stock issuance costs. The investor was also issued:
|
|
1)
|
Series I warrants to purchase 2,222,222 shares of common stock at a purchase price of $1.05 per share at any time before September 3, 2009;
|
|
2)
|
Series II warrants to purchase 1,866,666 shares of common stock at a purchase price of $1.25 per share at any time from December 3, 2009 to June 5, 2012; and
|
|
3)
|
Series III warrants to purchase 1,555,555 shares of common stock at a purchase price of $1.50 per share at any time from December 3, 2009 to June 5, 2014.
|
Gross Proceeds:
|
$ | 3,000,000 | ||
Allocated to liabilities:
|
||||
Warrant liabilities
|
3,451,194 | |||
Allocated to equity:
|
||||
Common stock and additional paid-in capital
|
- | |||
Allocated to expense:
|
||||
Financing expense
|
(122,257 | ) | ||
Derivative loss at inception
|
(328,937 | ) | ||
Total allocated to expense
|
(451,194 | ) | ||
Total allocated gross proceeds:
|
$ | 3,000,000 |
ad)
|
On June 9, 2009, the Company issued 1,833,341 shares of common stock and 862,246 warrants to purchase common stock at a purchase price of $1.05 per share to existing stockholders pursuant to the anti-dilution protection provisions of the private placements transacted on December 18, 2007 and March 20, 2008. The fair value of the additional warrants issued was approximately $422,300.
|
ae)
|
On September 4, 2009, an option holder exercised options to purchase shares of the Company’s common stock for cash of $3,600 and the Company issued an aggregate of 15,000 shares.
|
af)
|
On September 21, 2009, the Company issued 3,102,837 shares of common stock at a purchase price of $1.13 per share to an institutional investor for net proceeds of $3,371,340, which includes $128,659 of stock issuance costs.
|
13.
|
Common Stock (cont’d)
|
ag)
|
On October 23, 2009, the Company closed on a purchase agreement to issue 6,072,383 shares of common stock at a price of $0.82 per share to five institutional investors for gross proceeds of $5,000,000, which includes $351,928 of stock issuance costs. The investors were also issued warrants to purchase 2,125,334 shares of common stock at a purchase price of $1.00 per share, exercisable on or after the date of delivery until the five-year anniversary, and were recorded as liabilities at fair value. The closing costs included 245,932 warrants valued at $101,693 and were recorded as a financing expense.
|
Gross Proceeds:
|
$ | 5,000,000 | ||
Allocated to liabilities:
|
||||
Warrant liabilities
|
1,114,627 | |||
Allocated to equity:
|
||||
Common stock and additional paid-in capital
|
3,987,066 | |||
Allocated to expense:
|
||||
Financing expense
|
(101,693 | ) | ||
Total allocated gross proceeds:
|
$ | 5,000,000 |
ah)
|
On October 23, 2009, the Company issued 2,018,143 shares of common stock and 569,502 warrants to purchase common stock at a purchase price of $0.82 per share to existing stockholders pursuant to anti-dilution protection provisions of the private placements transacted on December 24, 2007 and March 20, 2008.The fair value of the additional warrants issued was approximately $476,200.
|
ai)
|
On February 12, 2010, the Company entered into two consulting agreements pursuant to which the Company issued 300,000 shares of common stock upon the execution of the agreements. Upon the extension of the term, 200,000 shares of common stock for each month will be issued until the termination of services.
|
Date of Issuance
|
Number of Shares Issued
|
Market Value Per Share
|
Total Market Value of Share Issuance
|
|||||||||
February 12, 2010
|
300,000 | $ | 1.22 | $ | 366,000 | |||||||
May 24, 2010
|
200,000 | 1.40 | 280,000 | |||||||||
June 15, 2010
|
200,000 | 1.15 | 230,000 | |||||||||
August 2, 2010
|
400,000 | 1.37 | 548,000 | |||||||||
September 21, 2010
|
200,000 | 1.20 | 240,000 | |||||||||
October 21, 2010
|
200,000 | 1.16 | 232,000 | |||||||||
November 11, 2010
|
200,000 | 1.06 | 212,000 | |||||||||
Total
|
1,700,000 | $ | 2,108,000 |
13.
|
Common Stock (cont’d)
|
aj)
|
In March 2010, warrant holders exercised their warrants to purchase shares of the Company’s common stock for cash of $1,297,001 and the Company issued an aggregate of 1,197,001 shares.
|
ak)
|
In March 2010, option holders exercised options to purchase shares of the Company’s common stock for cash of $21,240 and the Company issued an aggregate of 48,000 shares.
|
al)
|
In April 2010, warrant holders exercised their warrants to purchase shares of the Company’s common stock for cash of $1,966,375 and the Company issued an aggregate of 1,595,825 shares.
|
am)
|
On April 20, 2010, an option holder exercised options to purchase shares of the Company’s common stock for cash of $86,000 and the Company issued an aggregate of 107,500 shares.
|
an)
|
In May 2010, warrant holders exercised warrants to obtain shares of the Company’s common stock and the Company issued an aggregate of 547,674 shares.
|
ao)
|
On June 30, 2010, the Company entered into a purchase agreement to issue 6,666,667 shares of common stock at a price of $1.50 per share to investors for gross proceeds of $10,000,000, which includes $681,773 of stock issuance costs. The investors were also issued warrants to purchase 2,000,000 shares of common stock at an exercise price of $1.90 per share. The warrants became immediately exercisable on the date of delivery until the four-year anniversary of the date of issuance. These warrants were valued at $1,800,800 and recorded as warrant liabilities. The closing costs included 200,000 warrants valued at $180,080 and were recorded as a financing expense.
|
Gross Proceeds:
|
$ | 10,000,000 | ||
Allocated to liabilities:
|
||||
Warrant liabilities
|
1,980,880 | |||
Allocated to equity:
|
||||
Common stock and additional paid-in capital
|
8,199,200 | |||
Allocated to expense:
|
||||
Financing expense
|
(180,080 | ) | ||
Total allocated gross proceeds:
|
$ | 10,000,000 |
ap)
|
In November 2010, warrant holders exercised 936,883 cashless warrants to obtain shares of the Company’s common stock and the Company issued an aggregate of 247,491 shares.
|
aq)
|
In December 2010, warrant holders exercised 530,900 cashless warrants to obtain shares of the Company’s common stock and the Company issued an aggregate of 126,195 shares.
|
ar)
|
On January 19, 2011, the Company issued 2,334,515 shares of common stock at a purchase price of $1.69 per share to an institutional investor for net proceeds of $3,926,397, which includes $23,603 of stock issuance costs.
|
as)
|
On February 15, 2011, a warrant holder exercised warrants to purchase shares of the Company’s common stock for cash of $215,104 and the Company issued 209,042 shares.
|
at)
|
On February 28, 2011, an option holder exercised options to purchase shares of the Company’s common stock for cash of $6,000 and the Company issued 25,000 shares.
|
au)
|
On March 11, 2011, an option holder exercised options to purchase shares of the Company’s common stock for cash of $12,000 and the Company issued 50,000 shares.
|
13.
|
Common Stock (cont’d)
|
av)
|
On March 28, 2011, warrant holders exercised their warrants to purchase shares of the the Company’s common stock for cash of $102,857 and the Company issued 124,917 shares.
|
aw)
|
On March 31, 2011, the Company closed on a purchase agreement to issue 8,333,333 shares of common stock at a price of $1.20 per share to five institutional investors for gross proceeds of $10,000,000, which includes $803,791 of stock issuance costs. The investors were also issued warrants to purchase 3,333,333 shares of common stock at a purchase price of $1.50 per share, exercisable on or after six months after the closing date until the five-year anniversary of the initial exercise date, and were recorded as liabilities at fair value. The closing costs included 208,333 warrants valued at $97,667 and were recorded as a financing expense.
|
Gross Proceeds:
|
$ | 10,000,000 | ||
Allocated to liabilities:
|
||||
Warrant liabilities
|
2,924,333 | |||
Allocated to equity:
|
||||
Common stock and additional paid-in capital
|
7,173,334 | |||
Allocated to expense:
|
||||
Financing expense
|
(97,667 | ) | ||
Total allocated gross proceeds:
|
$ | 10,000,000 |
ax)
|
In September 2011, an option holder exercised options to purchase shares of the Company’s common stock for cash of $22,040 and the Company issued 28,000 shares.
|
14.
|
Stock-Based Compensation
|
14.
|
Stock-Based Compensation (cont’d)
|
Three Months Ended September 30,
|
Nine Months Ended September 30,
|
Cumulative from
March 19, 2001
(Inception) to
September 30,
|
||||||||||||||||||
2011
|
2010
|
2011
|
2010
|
2011
|
||||||||||||||||
Statement of operations line item: General and administrative:
|
||||||||||||||||||||
Payroll
|
$ | 138,170 | $ | 94,375 | $ | 397,192 | $ | 286,011 | $ | 2,390,708 | ||||||||||
Consulting and other professional fees
|
(16,915 | ) | (6,851 | ) | 30,265 | 81,961 | 790,220 | |||||||||||||
Research and development:
|
||||||||||||||||||||
Payroll
|
23,706 | 21,532 | 69,546 | 52,888 | 945,844 | |||||||||||||||
Consulting and other professional fees
|
(3,872 | ) | 2,546 | 16,252 | 14,445 | 1,325,505 | ||||||||||||||
Total
|
$ | 141,089 | $ | 111,602 | $ | 513,255 | $ | 435,305 | $ | 5,452,277 |
For the nine months ended September 30, 2011
|
||||||||||||
Date Granted
|
Number of Options Granted
|
Exercise Price
|
Grant Date Fair Value
|
|||||||||
February 7, 2011
|
130,000 | $ | 1.84 | $ | 180,326 | |||||||
June 6, 2011
|
100,000 | $ | 1.25 | 91,334 | ||||||||
June 10, 2011
|
20,000 | $ | 1.22 | 17,915 | ||||||||
September 8, 2011
|
150,000 | $ | 1.12 | 121,595 | ||||||||
Total
|
400,000 | $ | 411,170 | |||||||||
For the nine months ended September 30, 2010
|
||||||||||||
Date Granted
|
Number of Options Granted
|
Exercise Price
|
Grant Date Fair Value
|
|||||||||
February 17, 2010
|
375,000 | $ | 1.33 | $ | 304,043 | |||||||
June 14, 2010
|
160,000 | $ | 1.17 | 142,150 | ||||||||
September 17, 2010
|
190,000 | $ | 1.19 | 171,280 | ||||||||
Total
|
725,000 | $ | 617,473 |
14.
|
Stock-Based Compensation (cont’d)
|
Nine Months Ended September 30,
|
||||||||
2011
|
2010
|
|||||||
Black-Scholes weighted average assumptions
|
||||||||
Expected dividend yield
|
0 | % | 0 | % | ||||
Expected volatility
|
96-101 | % | 100-114 | % | ||||
Risk free interest rate
|
0.11-2.29 | % | 0.26-2.40 | % | ||||
Expected term (in years)
|
5 years
|
1- 5 years
|
2011
|
2010
|
|||||||||||||||
Number of Options
|
Weighted Avg. Exercise Price
|
Number of Options
|
Weighted Avg. Exercise Prices
|
|||||||||||||
Outstanding at January 1
|
8,076,795 | $ | 1.01 | 7,715,795 | $ | 0.98 | ||||||||||
Granted
|
400,000 | 1.39 | 725,000 | 1.26 | ||||||||||||
Exercised
|
(103,000 | ) | 0.39 | (155,500 | ) | 0.69 | ||||||||||
Cancelled
|
(192,000 | ) | 1.21 | (78,500 | ) | 1.00 | ||||||||||
Outstanding at September 30
|
8,181,795 | $ | 1.03 | 8,206,795 | $ | 1.02 |
14.
|
Stock-Based Compensation(cont’d)
|
Number of Options
|
Weighted Avg. Exercise Prices
|
Weighted Average Remaining Contractual Term
|
Aggregate Intrinsic Value
|
||||||||||
Outstanding at
September 30, 2011
|
8,181,795 | $ | 1.03 |
4.9 years
|
$ | 1,466,974 | |||||||
Exercisable at
September 30, 2011
|
6,971,795 | $ | 1.02 |
4.3 years
|
$ | 1,356,324 | |||||||
Outstanding at
December 31, 2010
|
8,076,795 | $ | 1.01 |
5.4 years
|
$ | 2,198,790 | |||||||
Exercisable at
December 31, 2010
|
6,762,795 | $ | 1.00 |
4.8 years
|
$ | 2,198,790 |
2011
|
||||||||
Number of Options
|
Weighted Average Fair Value at Grant Date
|
|||||||
Unvested at January 1, 2011
|
1,314,000 | $ | 0.77 | |||||
Granted
|
400,000 | $ | 1.03 | |||||
Vested
|
(415,000 | ) | $ | 0.85 | ||||
Cancelled
|
(89,000 | ) | $ | 0.90 | ||||
Unvested at September 30, 2011
|
1,210,000 | $ | 0.80 |
15.
|
Warrants
|
2011
|
2010
|
|||||||||||||||
Number of warrants
|
Weighted average exercise price
|
Number of warrants
|
Weighted average exercise price
|
|||||||||||||
Balance, January 1
|
5,624,583 | $ | 1.48 | 8,575,243 | $ | 1.10 | ||||||||||
Issued during the period
|
3,541,666 | $ | 1.50 | 2,200,000 | $ | 1.90 | ||||||||||
Exercised during the period
|
(333,959 | ) | $ | (0.95 | ) | (3,682,877 | ) | $ | (0.89 | ) | ||||||
Expired during the period
|
(156,148 | ) | $ | (0.82 | ) | - | $ | - | ||||||||
Balance, September 30
|
8,676,142 | $ | 1.53 | 7,092,366 | $ | 1.35 |
15.
|
Warrants (cont’d)
|
Fair Value as of:
|
||||||||||||
Warrant Issuance:
|
September 30, 2011
|
December 31, 2010
|
Transaction Date
|
|||||||||
December 18, 2007 financing
|
$ | - | $ | - | $ | 1,392,476 | ||||||
March 20, 2008 financing
|
- | 123,558 | 190,917 | |||||||||
June 5, 2009 financing:
|
||||||||||||
Series I warrants
|
- | - | 707,111 | |||||||||
Series II warrants
|
- | - | 1,315,626 | |||||||||
Series III warrants
|
485,800 | 751,022 | 1,306,200 | |||||||||
Warrants to placement agent
|
46,012 | 69,032 | 122,257 | |||||||||
October 23, 2009 financing:
|
||||||||||||
Warrants to institutional investors
|
579,650 | 694,377 | 1,012,934 | |||||||||
Warrants to placement agent
|
5,886 | 111,241 | 101,693 | |||||||||
June 30, 2010 financing
|
||||||||||||
Warrants to institutional investors
|
516,400 | 1,106,800 | 1,800,800 | |||||||||
Warrants to placement agent
|
28,040 | 110,680 | 180,080 | |||||||||
March 31, 2011 financing:
|
||||||||||||
Warrants to institutional investors
|
1,950,000 | - | 2,826,666 | |||||||||
Warrants to placement agent
|
41,918 | - | 97,667 | |||||||||
Total:
|
$ | 3,653,706 | $ | 2,966,710 | $ | 11,054,427 |
15.
|
Warrants (cont’d)
|
Number of Shares indexed as of:
|
||||||||||||
Warrant Issuance
|
September 30, 2011
|
December 31, 2010
|
Transaction Date
|
|||||||||
December 18, 2007 financing
|
- | - | 1,078,579 | |||||||||
March 20, 2008 financing
|
- | 281,065 | 128,572 | |||||||||
June 5, 2009 financing:
|
||||||||||||
Series I warrants
|
- | - | 2,222,222 | |||||||||
Series II warrants
|
- | - | 1,866,666 | |||||||||
Series III warrants
|
1,555,555 | 1,555,555 | 1,555,555 | |||||||||
Warrants to placement agent
|
132,143 | 132,143 | 142,857 | |||||||||
October 23, 2009 financing:
|
||||||||||||
Warrants to institutional investors
|
1,228,333 | 1,228,333 | 2,125,334 | |||||||||
Warrants to placement agent
|
18,445 | 227,487 | 245,932 | |||||||||
June 30, 2010 financing
|
||||||||||||
Warrants to institutional investors
|
2,000,000 | 2,000,000 | 2,000,000 | |||||||||
Warrants to placement agent
|
200,000 | 200,000 | 200,000 | |||||||||
March 31, 2011 financing:
|
||||||||||||
Warrants to institutional investors
|
3,333,333 | - | 3,333,333 | |||||||||
Warrants to placement agent
|
208,333 | - | 208,333 | |||||||||
Total:
|
8,676,142 | 5,624,583 | 15,107,383 |
December 18, 2007 financing:
|
September 30, 2011
|
December 31, 2010
|
Transaction Date
|
|||||||||
Trading market prices
|
$ | - | $ | - | $ | 1.75 | ||||||
Estimated future volatility
|
- | - | 143 | % | ||||||||
Dividend
|
- | - | - | |||||||||
Estimated future risk-free rate
|
- | - | 3.27 | % | ||||||||
Equivalent volatility
|
- | - | 106 | % | ||||||||
Equivalent risk-free rate
|
- | - | 3.26 | % | ||||||||
Estimated additional shares to be issued upon dilutive event
|
- | - | 98,838 |
March 20, 2008 financing:
|
September 30, 2011
|
December 31, 2010
|
Transaction Date
|
|||||||||
Trading market prices
|
$ | - | $ | 1.12 | $ | 2.14 | ||||||
Estimated future volatility
|
- | 75 | % | 142 | % | |||||||
Dividend
|
- | - | - | |||||||||
Estimated future risk-free rate
|
- | 0.47 | % | 1.95 | % | |||||||
Equivalent volatility
|
- | 42 | % | 97 | % | |||||||
Equivalent risk-free rate
|
- | 0.12 | % | 1.31 | % | |||||||
Estimated additional shares to be issued upon dilutive event
|
- | 25,462 | 7,479 |
15.
|
Warrants (cont’d)
|
June 5, 2009 financing:
|
September 30, 2011
|
December 31, 2010
|
Transaction Date
|
|||||||||
Trading market prices
|
$ | 1.00 | $ | 1.12 | $ | 1.14 | ||||||
Estimated future volatility
|
80-86 | % | 94-100 | % | 100 | % | ||||||
Dividend
|
- | - | - | |||||||||
Estimated future risk-free rate
|
0.76 | % | 1.84-4.18 | % | 0.63-4.31 | % | ||||||
Equivalent volatility
|
68 | % | 72-73 | % | 103-117 | % | ||||||